Molecule Details
InChIKeyBLTYWXMDJBDQPE-XHCALQHSSA-N
Canonical SMILESN#C[C@@H]1CCCN1C(=O)CNC(=O)c1ccnc2ccc(OCCCNC(=O)CCc3cn(CCOCCOCCOCCC(=O)N[C@@H](CCCCNC(=O)CCC(C(=O)O)N4CCCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)C4)C(=O)NCCCCC(=O)N(CCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O)Cc4ccc(Br)cc4)nn3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.5
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12884 FAP Homo sapiens Human PF00930 PF00326 8.8 IC50 BindingDB
Q04609 FOLH1 Homo sapiens Human PF02225 PF04389 PF04253 8.2 IC50 BindingDB