Molecule Details
InChIKeyBLMBNKDQXGINRE-UHFFFAOYSA-N
Compound Name4-(4-fluoro-3-((pyridin-2-ylmethyl)carbamoyl)phenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
Canonical SMILESCC1=C(C(=O)Nc2ccc3[nH]ncc3c2)C(c2ccc(F)c(C(=O)NCc3ccccn3)c2)NC(=O)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 8.0 IC50 ChEMBL;BindingDB
P25098 GRK2 Homo sapiens Human PF00169 PF00069 PF00615 6.8 IC50 ChEMBL;BindingDB
P34947 GRK5 Homo sapiens Human PF00069 PF00615 6.4 IC50 ChEMBL;BindingDB