Molecule Details
InChIKeyBKZIXMFZEWLONB-UHFFFAOYSA-N
Compound Name1-[6-(1,4-Diazepan-1-yl)-2-pyridinyl]-6-(5-propan-2-yl-3-pyridinyl)pyrazolo[4,3-c]pyridine
Canonical SMILESCC(C)c1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCCNCC3)n2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.75
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 10.5 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 10.2 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.6 Ki ChEMBL;BindingDB