Molecule Details
InChIKeyBKOOLLRJJOFPDK-UHFFFAOYSA-N
Canonical SMILESCC(C)c1c2sc(-c3nc(Nc4ccc(C5CCN(C)CC5)cn4)ncc3F)cc2nn1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24385 CCND1 Homo sapiens Human PF02984 PF00134 7.0 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.0 IC50 ChEMBL