Molecule Details
InChIKeyBJWFIOSIGHDXLF-QBHOUYDASA-N
Compound Name(2S)-2-[(1-{[3-cyclohexyl-1-(1,3-thiazol-5-yl)propoxy]carbonyl}-5-(2-methylphenyl)-1,2,3,6-tetrahydropyridin-4-yl)formamido]-4-(methylsulfanyl)butanoic acid
Canonical SMILESCSCC[C@H](NC(=O)C1=C(c2ccccc2C)CN(C(=O)OC(CCC2CCCCC2)c2cncs2)CC1)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.15
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.2 IC50 ChEMBL