Molecule Details
InChIKeyBJBQASWPUALPOY-UHFFFAOYSA-N
Compound Name5-chloro-4-[(5-chloro-6-cyclopropylpyridin-3-yl)oxy]-2-fluoro-N-(methanesulfonyl)benzamide
Canonical SMILESCS(=O)(=O)NC(=O)c1cc(Cl)c(Oc2cnc(C3CC3)c(Cl)c2)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15858 SCN9A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.5 IC50 ChEMBL;BindingDB
O60939 SCN2B Homo sapiens Human PF07686 7.3 IC50 ChEMBL
Q07699 SCN1B Homo sapiens Human PF07686 7.3 IC50 ChEMBL