Molecule Details
InChIKeyBJACFZCSEUDRAZ-UHFFFAOYSA-N
Compound Name4-methoxy-N-(6-methoxy-3-pyridinyl)-N-[[5-(2-methylphenyl)-2-pyridinyl]methyl]benzenesulfonamide
Canonical SMILESCOc1ccc(S(=O)(=O)N(Cc2ccc(-c3ccccc3C)cn2)c2ccc(OC)nc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.6
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30559 OXTR Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P37288 AVPR1A Homo sapiens Human PF00001 PF08983 7.8 Ki ChEMBL;BindingDB
P30518 AVPR2 Homo sapiens Human PF00001 6.6 Ki ChEMBL;BindingDB