Molecule Details
InChIKeyBJABGWNNTUGRHH-LRXLXLKKSA-N
Canonical SMILESCOc1ccc(CCNC(=O)C(C)(Cc2c[nH]c3ccccc23)NC(=O)OC2[C@H]3C[C@@H]4C[C@@H](C[C@H]2C4)C3)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.94
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.9 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.9 Ki ChEMBL