Molecule Details
InChIKeyBIMJVPXBEXJSPH-YTTGMZPUSA-N
Compound Name3-[(4-cyclohexylpiperazin-1-yl)methyl]-2-phenyl-N-[(1S)-1-phenylpropyl]quinoline-4-carboxamide
Canonical SMILESCC[C@H](NC(=O)c1c(CN2CCN(C3CCCCC3)CC2)c(-c2ccccc2)nc2ccccc12)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29371 TACR3 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P21452 TACR2 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB