Molecule Details
InChIKeyBIJXMFDKONGOAN-UHFFFAOYSA-N
Compound Name1-[N'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)phenyl]carbamimidoyl]-3-[6-[[N'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)phenyl]carbamimidoyl]carbamoylamino]hexyl]urea
Canonical SMILESCc1nc(N)sc1-c1ccc(N/C(N)=N/C(=O)NCCCCCCNC(=O)/N=C(\N)Nc2ccc(-c3sc(N)nc3C)cc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5N1 HRH3 Homo sapiens Human PF00001 8.5 Kd ChEMBL
P35367 HRH1 Homo sapiens Human PF00001 8.3 Kd ChEMBL
Q9H3N8 HRH4 Homo sapiens Human PF00001 7.8 Kd ChEMBL
P25021 HRH2 Homo sapiens Human PF00001 7.2 Kd ChEMBL