Molecule Details
InChIKeyBIIBGRGPRSJNLG-KWLHPURYSA-N
Canonical SMILESCOc1cc(N[C@H]2CCc3c(-c4cccc(-c5ccc(CNC[C@@H]6CCC(=O)N6)c(OC)n5)c4Cl)cccc32)c(Cl)cc1CN1CC[C@@](C)(C(=O)O)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL10.19
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15116 PDCD1 Homo sapiens Human PF07686 10.2 IC50 ChEMBL;BindingDB
Q9NZQ7 CD274 Homo sapiens Human PF08205 PF07686 10.2 IC50 ChEMBL