Molecule Details
InChIKeyBIABSXPPEYWVER-UHFFFAOYSA-N
Compound Name1-[(6-Bromanyl-1,3-Benzodioxol-5-Yl)methyl]-4-Chloranyl-Pyrazolo[3,4-D]pyrimidin-6-Amine
Canonical SMILESNc1nc(Cl)c2cnn(Cc3cc4c(cc3Br)OCO4)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12931 TRAP1 Homo sapiens Human PF13589 PF00183 7.0 IC50 ChEMBL;BindingDB
P14625 HSP90B1 Homo sapiens Human PF13589 PF00183 6.3 IC50 ChEMBL;BindingDB
P07900 HSP90AA1 Homo sapiens Human PF13589 PF00183 6.3 IC50 ChEMBL;BindingDB