Molecule Details
InChIKeyBHHVWPMBOQGGMM-UHFFFAOYSA-N
Compound Name2-[2-(cyclopropanecarbonylamino)-4-pyridinyl]-4-methoxy-N-[6-(1,2,3,4-tetrahydroacridin-9-ylamino)hexyl]-1,3-thiazole-5-carboxamide
Canonical SMILESCOc1nc(-c2ccnc(NC(=O)C3CC3)c2)sc1C(=O)NCCCCCCNc1c2c(nc3ccccc13)CCCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P22303 ACHE Homo sapiens Human PF08674 PF00135 7.7 IC50 ChEMBL;BindingDB
P06276 BCHE Homo sapiens Human PF08674 PF00135 7.0 IC50 ChEMBL;BindingDB