Molecule Details
InChIKeyBGNRMTUXZUCPDO-AWEZNQCLSA-N
Compound Name5-[3-(2-fluorophenyl)-1H-indol-5-yl]-N-[(3S)-piperidin-3-yl]-1,3,4-thiadiazol-2-amine
Canonical SMILESFc1ccccc1-c1c[nH]c2ccc(-c3nnc(N[C@H]4CCCNC4)s3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB