Molecule Details
InChIKeyBGNDQDYZQSRSAU-UHFFFAOYSA-N
Compound Name3-[2-(Pyridin-4-yl)-1,3-thiazol-4-yl]-1,2,3,4-tetrahydroquinazolin-2-one
Canonical SMILESO=C1Nc2ccccc2CN1c1csc(-c2ccncc2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.02
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00535 CDK5 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
Q15078 CDK5R1 Homo sapiens Human PF03261 7.1 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.8 IC50 BindingDB