Molecule Details
InChIKeyBGJDVOKZOHLJPT-UHFFFAOYSA-N
Compound Name3-(1,2,3,4-Tetrahydroisoquinoline-2-yl)methyl-1H-pyrrolo[2,3-b]pyridine
Canonical SMILESc1ccc2c(c1)CCN(Cc1c[nH]c3ncccc13)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB