Target not found.
Molecule Details
InChIKeyBFJGLGUWQKURET-IBGZPJMESA-N
Compound Name(S)-7-(4-fluorophenyl)-8-(3-methylimidazo[1,2-a] pyridin-6-yl)-2-((l-methylpyrrolidin-2-yl)methyl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-amine
Canonical SMILESCc1cnc2ccc(-c3c(-c4ccc(F)cc4)nc(N)n4nc(C[C@@H]5CCCN5C)nc34)cn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.5 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.2 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB