Molecule Details
InChIKeyBENOEPUDOPGLCP-XMMPIXPASA-N
Compound Name5-[(5R)-5-[(7-fluoro-1,1-dimethyl-2,3-dihydro-1H-inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5H)-yl]-5-oxopentanoic acid
Canonical SMILESCOc1ccc2c(n1)CCN(C(=O)CCCC(=O)O)[C@H]2C(=O)Nc1cc(F)c2c(c1)CCC2(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL9.1
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9HBA0 TRPV4 Homo sapiens Human PF00023 PF00520 9.7 IC50 BindingDB
P51449 RORC Homo sapiens Human PF00104 PF00105 8.5 IC50 ChEMBL;BindingDB