Molecule Details
InChIKeyBDLXCRNZHKNUCS-VFNWGFHPSA-N
Compound Name2-[3-(4-Benzyloxy-phenyl)-3-methyl-2-oxo-pyrrolidin-1-yl]-N-hydroxy-propionamide
Canonical SMILESC[C@H](C(=O)NO)N1CC[C@@](C)(c2ccc(OCc3ccccc3)cc2)C1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.89
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 8.4 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.7 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 7.5 Ki ChEMBL;BindingDB