Molecule Details
InChIKeyBDDQTHYDKKYXON-UHFFFAOYSA-N
Compound NameUS9890185, Example 38(o)
Canonical SMILESCOc1c(CC(N)=O)cc(C(C)(C)C)cc1NC(=O)Nc1ccc(Oc2ccnc(Nc3ccn(C)n3)c2)c2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 7.3 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 6.4 IC50 ChEMBL;BindingDB