Molecule Details
InChIKeyBCWROVBBUOSFGD-UHFFFAOYSA-N
Compound Name2-((1H-imidazol-2-yl)methylthio)-6-amino-4-(4-methoxyphenyl)pyridine-3,5-dicarbonitrile
Canonical SMILESCOc1ccc(-c2c(C#N)c(N)nc(SCc3ncc[nH]3)c2C#N)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 7.6 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB