Molecule Details
InChIKeyBCRJIIJVFJJYRD-UHFFFAOYSA-N
Compound Name4-tert.-butyl-N-[6-(3-(2-thiophenesulfonylamino)-propoxy)-5-(o-methoxyphenoxy)-2-cyclopropyl-4-pyrimidinyl]-benzene-sulfonamide
Canonical SMILESCOc1ccccc1Oc1c(NS(=O)(=O)c2ccc(C(C)(C)C)cc2)nc(C2CC2)nc1OCCCNS(=O)(=O)c1cccs1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 8.7 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB