Molecule Details
InChIKeyBBVNYSAAUUALLQ-UHFFFAOYSA-N
Compound Name6-[(Naphthalen-1-ylamino)methyl]pyrido[2,3-d]pyrimidine-2,4-diamine
Canonical SMILESNc1nc(N)c2cc(CNc3cccc4ccccc34)cnc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.1 IC50 ChEMBL;BindingDB
P0ABQ4 folA Escherichia coli (strain K12) Pathogen PF00186 7.1 IC50 ChEMBL;BindingDB
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 6.8 IC50 ChEMBL;BindingDB