Molecule Details
InChIKeyBBDWOHDPFZUDCG-INIZCTEOSA-N
Compound Name(S)-benzyl 1-(4-tert-butylthiazol-2-ylamino)-1-oxo-6-(sulfamoylamino)hexan-2-ylcarbamate
Canonical SMILESCC(C)(C)c1csc(NC(=O)[C@H](CCCCNS(N)(=O)=O)NC(=O)OCc2ccccc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.08
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 6.1 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.1 pIC50 TTD_MultiTarget
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.1 IC50 ChEMBL;BindingDB