Molecule Details
InChIKeyAZJKTFMVKCDMSG-JTQLQIEISA-N
Compound NameVrk1/CK1-IN-1
Canonical SMILESCc1cc(CN2C(=O)[C@H](C)N(C)c3nc(Nc4cc(F)c(O)c(F)c4)ncc32)on1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.42
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P49674 CSNK1E Homo sapiens Human PF00069 8.1 Ki ChEMBL
P48730 CSNK1D Homo sapiens Human PF00069 8.1 Ki ChEMBL
Q99986 VRK1 Homo sapiens Human PF00069 7.4 Ki ChEMBL
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 6.1 Ki ChEMBL