Molecule Details
InChIKeyAZHXFKCTCUPFGL-UHFFFAOYSA-N
Compound Name4-({4-[(2-Fluoro-5-methylphenyl)amino]pyrimidin-2-yl}amino)benzene-1-sulfonamide
Canonical SMILESCc1ccc(F)c(Nc2ccnc(Nc3ccc(S(N)(=O)=O)cc3)n2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.22
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 8.2 pIC50 TTD_MultiTarget
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 8.2 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 8.2 pIC50 TTD_MultiTarget