Molecule Details
InChIKeyAZCHQQLGTDJHFL-ZDUSSCGKSA-N
Compound Name4-N-(5-ethyl-1H-pyrazol-3-yl)-2-N-[(1S)-1-(5-fluoro-2-pyridinyl)ethyl]-5-methylquinazoline-2,4-diamine
Canonical SMILESCCc1cc(Nc2nc(N[C@@H](C)c3ccc(F)cn3)nc3cccc(C)c23)n[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43250 GRK6 Homo sapiens Human PF00069 PF00615 7.1 IC50 ChEMBL;BindingDB
P08069 IGF1R Homo sapiens Human PF00757 PF07714 PF01030 6.8 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB