Molecule Details
InChIKeyAYVATFZLZLWIPA-UHFFFAOYSA-N
Compound Name5-[4-(3,3-dimethylpiperazin-1-yl)phenyl]-2-(3-methyl-1H-indol-4-yl)-1,3-oxazole-4-carboxamide
Canonical SMILESCc1c[nH]c2cccc(-c3nc(C(N)=O)c(-c4ccc(N5CCNC(C)(C)C5)cc4)o3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 9.3 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 7.8 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB