Molecule Details
InChIKeyAYOYRQBAZIBAOY-UHFFFAOYSA-N
Compound Name7-[3-[4-(2-methoxyphenyl)piperazin-1-yl]propoxy]-1H-quinolin-2-one
Canonical SMILESCOc1ccccc1N1CCN(CCCOc2ccc3ccc(=O)[nH]c3c2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB