Molecule Details
InChIKeyAYNCNNOVAOFEMG-YZVOILCLSA-N
Compound NameN-[4-[(3S,4S,5R)-3-amino-4-cyano-5-methylpiperidin-1-yl]-3-pyridinyl]-6-(2,6-difluoro-4-methylphenyl)-5-fluoropyridine-2-carboxamide
Canonical SMILESCc1cc(F)c(-c2nc(C(=O)Nc3cnccc3N3C[C@@H](N)[C@@H](C#N)[C@@H](C)C3)ccc2F)c(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.68
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.9 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB