Molecule Details
InChIKeyAXKZEVVSSSVTOD-UHFFFAOYSA-N
Compound Name4-{3-[5-(piperidin-1-ylmethyl)-1H-indol-2-yl]-1H-indazol-6-yl}-1,2-thiazole
Canonical SMILESc1cc2[nH]c(-c3n[nH]c4cc(-c5cnsc5)ccc34)cc2cc1CN1CCCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.8
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14757 CHEK1 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
P50613 CDK7 Homo sapiens Human PF00069 7.8 IC50 ChEMBL
P51946 CCNH Homo sapiens Human PF16899 PF00134 7.7 IC50 BindingDB