Molecule Details
InChIKeyAXBBWELSCMNUPM-UHFFFAOYSA-N
Compound NameN-Hydroxy-N-{1-(4-hydroxyimino-cyclohexylmethyl)-2-[4-(2-methyl-quinolin-4-ylmethoxy)-benzenesulfonyl]-ethyl}-formamide
Canonical SMILESCc1cc(COc2ccc(S(=O)(=O)CC(CC3CCC(N=O)CC3)N(O)C=O)cc2)c2ccccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.09
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P78536 ADAM17 Homo sapiens Human PF16698 PF00200 PF13574 8.5 IC50 BindingDB
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 6.5 IC50 BindingDB
P08254 MMP3 Homo sapiens Human PF00045 PF00413 PF01471 6.3 IC50 BindingDB