Target not found.
Molecule Details
InChIKeyAWTKTGLFVCACHC-UHFFFAOYSA-N
Compound Name4-[(5-chloro-4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]-N-ethylpiperidine-1-carboxamide
Canonical SMILESCCNC(=O)N1CCC(Nc2ncc(Cl)c(-c3cnc4ccccn34)n2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.96
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.2 pIC50 TTD_MultiTarget