Molecule Details
InChIKeyAWLFNVKRXDPUCZ-QFIPXVFZSA-N
Compound Name(S)-2-(4-(dimethylamino)benzamido)-N8-hydroxy-N1-(quinolin-8-yl)octanediamide
Canonical SMILESCN(C)c1ccc(C(=O)N[C@@H](CCCCCC(=O)NO)C(=O)Nc2cccc3cccnc23)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.13
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 7.7 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 7.7 pIC50 TTD_MultiTarget
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.0 IC50 ChEMBL;BindingDB