Molecule Details
InChIKeyAWEQRQAMCRCOJY-INIZCTEOSA-N
Compound Name(S)-1-(6-(3-methylpiperazin-1-yl)pyridin-2-yl)-6-(5-(oxetan-3-yl)pyridin-3-yl)-1H-pyrazolo[4,3-c]pyridine
Canonical SMILESC[C@H]1CN(c2cccc(-n3ncc4cnc(-c5cncc(C6COC6)c5)cc43)n2)CCN1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 10.0 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.7 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.0 Ki ChEMBL;BindingDB