Molecule Details
InChIKeyAVHWMAVUUHFRKE-UAVUOLJFSA-N
Canonical SMILESO=C(O)[C@H]1CC[C@H](C(=O)N2CC[C@](c3ccc(C(F)(C(F)(F)F)C(F)(F)F)cc3)(S(=O)(=O)c3ccc(F)cc3)C2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P51449 RORC Homo sapiens Human PF00104 PF00105 7.3 IC50 ChEMBL;BindingDB
P10632 CYP2C8 Homo sapiens Human PF00067 6.2 IC50 ChEMBL