Molecule Details
InChIKeyATSRNUWJDQUCNU-UHFFFAOYSA-N
Compound Name1-[3-Tert-butyl-1-(4-methylphenyl)pyrazol-5-yl]-3-[4-[2-[2-(methylcarbamoylamino)-4-pyridinyl]ethoxy]naphthalen-1-yl]urea
Canonical SMILESCNC(=O)Nc1cc(CCOc2ccc(NC(=O)Nc3cc(C(C)(C)C)nn3-c3ccc(C)cc3)c3ccccc23)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P08631 HCK Homo sapiens Human PF07714 PF00017 PF00018 7.6 IC50 ChEMBL;BindingDB
P53778 MAPK12 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB