Molecule Details
InChIKeyASXDLQKYJZCCLE-UHFFFAOYSA-N
Compound Name4-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1H-indol-3-yl]-2-Pyridinamine
Canonical SMILESNc1cc(-c2c[nH]c3ccc(-c4nnc(N)s4)cc23)ccn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.74
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB