Molecule Details
InChIKeyASUWZCFQGVUVGX-UHFFFAOYSA-N
Compound Name4-[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-piperazine-1-carboxylic acid 2-(2,2,2-trifluoro-ethyl)-benzyl ester
Canonical SMILESN#Cc1ccc(Cn2cncc2CN2CCN(C(=O)OCc3ccccc3CC(F)(F)F)CC2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.74
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.1 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.8 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 8.3 IC50 ChEMBL