Molecule Details
InChIKeyASUAOIWGQADQOH-PYPSSTHSSA-N
Compound NameAc-YK[CEHdFRWC]-NH2
Canonical SMILESCC(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H]1CSSC[C@H](C(N)=O)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2c[nH]cn2)NC(=O)[C@@H](CCC(=O)O)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P32245 MC4R Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
Q01726 MC1R Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB