Molecule Details
InChIKeyASLFQIAAFMLPFR-PBHICJAKSA-N
Compound Name3-(furo[3,2-d]pyrimidin-4-ylamino)-6,6-dimethyl-N-[(1S,2R)-2-phenylcyclopropyl]-1,4-dihydropyrrolo[3,4-d]pyrazole-5-carboxamide
Canonical SMILESCC1(C)c2[nH]nc(Nc3ncnc4ccoc34)c2CN1C(=O)N[C@H]1C[C@@H]1c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35372 OPRM1 Homo sapiens Human PF00001 7.2 Ki ChEMBL
P41143 OPRD1 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
O96013 PAK4 Homo sapiens Human PF00786 PF00069 7.2 Ki ChEMBL;BindingDB