Molecule Details
InChIKeyASAZVVSUHCMYAU-UHFFFAOYSA-N
Compound Name3-(2-amino-1H-benzimidazol-4-yl)-6-(2-aminoethylsulfonyl)-2-(2H-tetrazol-5-yl)benzenesulfonamide
Canonical SMILESNCCS(=O)(=O)c1ccc(-c2cccc3nc(N)[nH]c23)c(-c2nn[nH]n2)c1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.38
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.6 IC50 ChEMBL;BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.4 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.1 IC50 BindingDB