Molecule Details
InChIKeyAQSNIXKAKUZPSI-SSTWWWIQSA-N
Compound NameStx-140
Canonical SMILESCOc1cc2c(cc1OS(N)(=O)=O)CC[C@@H]1[C@@H]2CC[C@]2(C)[C@@H](OS(N)(=O)=O)CC[C@@H]12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB08416
Drug Name(9BETA,13ALPHA,14BETA,17ALPHA)-2-METHOXYESTRA-1,3,5(10)-TRIENE-3,17-DIYL DISULFAMATE
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 50200936 CHEMBL218382 ChemSpider: 7980062 PDB: PO1 PubChem:9804302 PubChem:99444887 ZINC: ZINC000003975451
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08842 STS Homo sapiens Human PF00884 PF14707 7.4 IC50 ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.7 Kd ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.4 IC50 ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P00918 CA2 Carbonic anhydrase 2 inhibitor targets
P08842 STS Steryl-sulfatase inhibitor targets