Molecule Details
InChIKeyAQSMXTCYTUNCFB-UHFFFAOYSA-N
Compound Name7-(2-cyclohexylethyl)-6-((pyridin-2-yloxy)methyl)-7H-pyrrolo[2,3-d]pyrimidine-2-carbonitrile
Canonical SMILESN#Cc1ncc2cc(COc3ccccn3)n(CCC3CCCCC3)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25774 CTSS Homo sapiens Human PF08246 PF00112 8.0 IC50 ChEMBL;BindingDB
P43235 CTSK Homo sapiens Human PF08246 PF00112 6.6 IC50 ChEMBL;BindingDB
P07711 CTSL Homo sapiens Human PF08246 PF00112 6.1 IC50 ChEMBL;BindingDB