Molecule Details
InChIKeyAQGNHMOJWBZFQQ-UHFFFAOYSA-N
Canonical SMILESCc1cnc(-c2cnc(NCCNc3ccc(C#N)cn3)nc2-c2ccc(Cl)cc2Cl)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB19676
Drug NameLaduviglusib
CAS Number252917-06-9
Groups experimental
ATC Codes nan
DescriptionLaduviglusib is a small molecule drug. Laduviglusib has a monoisotopic molecular weight of 464.1 Da.

Categories: Glycogen Synthase Kinase 3, antagonists & inhibitors
Cross-references: BindingDB: 50325983 ChEBI: 91091 CHEMBL412142 PDB: 65C ZINC: ZINC000029053046
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P49840 GSK3A Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
DrugBank Target Actions (4)
Target Gene Target Name Action Type
P06493 CDK1 Cyclin-dependent kinase 1 inhibitor targets
P28482 MAPK1 Mitogen-activated protein kinase 1 inhibitor targets
P49840 GSK3A Glycogen synthase kinase-3 alpha inhibitor targets
P49841 GSK3B Glycogen synthase kinase-3 beta inhibitor targets