Molecule Details
InChIKeyAQFMGFCVDBEMQE-UHFFFAOYSA-N
Compound NameN-[3-[[4-[3-(cyclopropanecarbonylamino)propylamino]-5-iodopyrimidin-2-yl]amino]phenyl]pyrrolidine-1-carboxamide
Canonical SMILESO=C(NCCCNc1nc(Nc2cccc(NC(=O)N3CCCC3)c2)ncc1I)C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 7.2 IC50 ChEMBL;BindingDB
O75385 ULK1 Homo sapiens Human PF12063 PF21127 PF00069 7.2 IC50 ChEMBL;BindingDB
Q8IYT8 ULK2 Homo sapiens Human PF12063 PF21127 PF00069 6.7 IC50 ChEMBL;BindingDB