Molecule Details
InChIKeyAPWGKQAYROBBCL-UHFFFAOYSA-N
Compound Name[2-Amino-3-[(2,6-difluorophenyl)methyl]benzimidazol-5-yl]-(2-chloro-6-fluorophenyl)methanone
Canonical SMILESNc1nc2ccc(C(=O)c3c(F)cccc3Cl)cc2n1Cc1c(F)cccc1F
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.31
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.5 pIC50 TTD_MultiTarget
P06493 CDK1 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget
P11802 CDK4 Homo sapiens Human PF00069 7.2 pIC50 TTD_MultiTarget