Molecule Details
InChIKeyAPNJYYQXBHETAR-UHFFFAOYSA-N
Compound Name7,8-Dimethoxy-3-(4-quinolin-6-ylmethyl-piperazin-1-ylmethyl)-3a,4-dihydro-3H-chromeno[4,3-c]isoxazole
Canonical SMILESCOc1cc2c(cc1OC)C1=NOC(CN3CCN(Cc4ccc5ncccc5c4)CC3)C1CO2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18825 ADRA2C Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P08913 ADRA2A Homo sapiens Human PF00001 6.9 Ki ChEMBL;BindingDB
P18089 ADRA2B Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB