Molecule Details
InChIKeyAPKPENVZICKJOY-UHFFFAOYSA-N
Canonical SMILESc1ccc2c(c1)c1cnc(Nc3ccc(N4CCNCC4)nn3)nc1n2C1CCCC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.01
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00534 CDK6 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB