Molecule Details
InChIKeyAPIFLWWBMVHSHA-KRWDZBQOSA-N
Compound Name(13aS)-12-bromo-3-methoxy-9-propoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinoline-2,10-diol
Canonical SMILESCCCOc1c(O)cc(Br)c2c1CN1CCc3cc(OC)c(O)cc3[C@@H]1C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21728 DRD1 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB